Bilaid C1

Bilaid C1

$263.00 - 1 mg

$921.00 - 5 mg

All prices in Australian dollars

CAS #
2393866-15-2
Molecular Formula
C28H39N5O5
Molecular Weight
525.64
Purity
>95% by HPLC
Long Term Storage
-20°C
Solubility
Soluble in methanol or DMSO
Clear

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Application Notes

Bilaid C1 (YvVf-NH2) is the semi-synthetic analogue of Bilaid C, an unusual tetrapeptide isolated from an Australian estuarine isolate of Penicillium sp. MST-MF667. Conversion of the terminal carboxylate to its corresponding amide enhanced the μ-​opioid agonist potency leading to the design of more potent analogues, bilorphin and bilactorphin.

References

  • A tetrapeptide class of biased analgesics from an Australian fungus targets the μ-​opioid receptor. Dekan Z et al. Proc Nat Acad Sci. 2019, 116, 22535.

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