Bilaid B1

Bilaid B1

$280.00 - 1 mg

$980.00 - 5 mg

All prices in Australian dollars

Code
BIA-B2277
CAS #
2393866-07-2
Molecular Formula
C28H39N5O5
Molecular Weight
525.64
Purity
>95% by HPLC
Long Term Storage
-20°C
Solubility
Soluble in methanol or DMSO

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Application Notes

Bilaid B1 (FvVy-NH2) is the semi-synthetic analogue of Bilaid B, an unusual tetrapeptide isolated from an Australian estuarine isolate of Penicillium sp. MST-MF667. Conversion of the terminal carboxylate to its corresponding amide enhanced the μ-​opioid agonist potency leading to the design of more potent analogues, bilorphin and bilactorphin.

References

  • A tetrapeptide class of biased analgesics from an Australian fungus targets the μ-​opioid receptor. Dekan Z. et al. Proc Nat Acad Sci. 2019, 116, 22535.

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