Bilaid C

Bilaid C

$263.00 - 1 mg

$921.00 - 5 mg

All prices in Australian dollars

CAS #
2393866-13-0
Molecular Formula
C28H38N4O6
Molecular Weight
526.62
Purity
>95% by HPLC
Long Term Storage
-20°C
Solubility
Soluble in methanol or DMSO
Clear

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Application Notes

Bilaid C (YvVf-OH) is a hydroxylated analogue of a family of tetrapeptides with an unusual alternating LDLD chirality isolated from an Australian estuarine isolate of Penicillium sp. MST-MF667. Bilaid C is an isomer of bilaid A with terminal L-phenylalanine and D-tyrosines inverted to their D and L-isomers. Bilaid C exhibited very weak μ-​opioid agonist and the class formed the foundation for the design of more potent analogues, bilorphin and bilactorphin. The bioassay profile of bilaid C has not been extensively investigated.

References

  • A tetrapeptide class of biased analgesics from an Australian fungus targets the μ-​opioid receptor. Dekan Z. et al. Proc Nat Acad Sci. 2019, 116, 22535.

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