Bilaid A
Bilaid A
$263.00 - 1 mg
$921.00 - 5 mg
All prices in Australian dollars
- CAS #
- NA
- Molecular Formula
- C28H38N4O5
- Molecular Weight
- 510.6
- Purity
- >95% by HPLC
- Long Term Storage
- -20°C
- Solubility
- Soluble in methanol or DMSO
Download Data Sheets
Application Notes
The bilaids are tetrapeptides with an unusual alternating LDLD chirality isolated from an Australian estuarine isolate of Penicillium sp.. Bilaids are weak μ-opioid agonists (Ki = 3.1 µM using HEK293 cell membranes expressing the human receptor) that inhibit forskolin-induced cAMP accumulation in HEK293 cells expressing the human µ-opioid receptor by 21% when used at a concentration of 10 µM.
References
- A tetrapeptide class of biased analgesics from an Australian fungus targets the μ-opioid receptor. Dekan Z et al. Proc Nat Acad Sci 2019, 116, 22535.
Other Products
Related products
-
Ansatrienin A
$155.00 – $543.00CAS #: 82189-03-5View Product
Molecular Formula: C36H48N2O8
Molecular Weight: 636.8 -
Anhydroophiobolin A
$287.00 – $1,005.00CAS #: 6026-65-9View Product
Molecular Formula: C25H34O3
Molecular Weight: 382.5 -
Hydroxyoligomycin A, 21-
$287.00 – $1,005.00CAS #: 102042-09-1View Product
Molecular Formula: C45H74O12
Molecular Weight: 807.1
